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OncoMatch/Clinical Trials/NCT07114601

A Study of LY4257496 in Participants With Cancer (OMNIRAY)

Is NCT07114601 recruiting? Yes, currently enrolling (Jun 2026). This Phase 1 trial studies multiple treatments including LY4257496 and Standard of Care Anticancer Therapies for breast neoplasms.

Phase 1RecruitingEli Lilly and CompanyNCT07114601Data as of Jun 2026Location: International · 7 countries

Treatment: LY4257496 · Standard of Care Anticancer TherapiesThe main purpose of this study is to evaluate safety, tolerability, and efficacy of LY4257496 alone and as part of relevant standard of care (SOC) combination therapy in participants with Gastrin-releasing Peptide Receptor (GRPR)-positive advanced breast, colorectal, prostate, and endometrial cancer. The study will also evaluate the safety, tolerability, and efficacy of LY4257529 to identify cancer with high levels of a protein called GRPR. This is a 2-part study. Participation could last up to 36 weeks or until your tumor progresses.

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Extracted eligibility criteria

Treatments studied

Other

LY4257496Standard of Care Anticancer Therapies

Cancer type

Breast Carcinoma

Colorectal Cancer

Endometrial Cancer

Biomarker criteria

Required: GRPR positive

Must have GRPR-positive disease, defined by investigator assessment of GRPR imaging.

Required: ESR1 expression (positive)

To fulfill the requirement for ER+ disease by local testing, a tumor must express the ER immunohistochemistry, as defined in the relevant American Society of Clinical Oncology (ASCO)/College of American Pathologists (CAP) guidelines.

Required: HER2 (ERBB2) expression

HER2 status should be determined by local testing, as defined in the relevant ASCO/CAP Guidelines.

Performance status

ECOG 0–1(Restricted strenuous activity)

Prior therapy

Cannot have received: radiopharmaceutical or radioligand therapy

Exception: Phase 1a (Cohort A1 and A2) only; prior ¹⁷⁷Lu-PSMA-617 permitted for mCRPC

Phase 1a (Cohort A1 and A2) only: Previously received radiopharmaceutical or radioligand therapy. For participants with metastatic castration-resistant prostate cancer (mCRPC), prior ¹⁷⁷Lu-prostate-specific membrane antigen (PSMA)-617 is permitted.

Cannot have received: hemi-body or whole-body radiotherapy

Previously received any prior hemi-body or whole-body radiotherapy

Cannot have received: external beam radiation therapy to >25% of bone marrow

prior external beam radiation therapy (EBRT) to greater than 25% of the bone marrow

Structured fields extracted by AI. May contain errors — verify against the official protocol.

US trial sites

  • City of Hope · Duarte, California
  • University of California, Los Angeles (UCLA) · Santa Monica, California
  • Stanford University Medical Center · Stanford, California
  • Biogenix Molecular, LLC · Miami, Florida
  • Moffitt · Tampa, Florida

Showing up to 5 US sites.

See all sites on ClinicalTrials.gov →

Frequently asked questions

Is NCT07114601 currently recruiting?

Yes, this trial is currently recruiting patients.

Are there prior therapy exclusions?

Yes. Prior radiopharmaceutical or radioligand therapy, hemi-body or whole-body radiotherapy, external beam radiation therapy to >25% of bone marrow disqualifies patients from enrollment.

Does this trial require GRPR?

Yes, GRPR positive is a required biomarker for enrollment.

Does this trial require ESR1?

Yes, ESR1 expression is a required biomarker for enrollment.

Does this trial require ERBB2?

Yes, ERBB2 expression is a required biomarker for enrollment.

Could you qualify for this trial?

Enter your biomarker results to see how this trial's eligibility criteria match your specific cancer profile.

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