OncoMatch

OncoMatch/Clinical Trials/NCT04300556

A Study to Evaluate the Safety, Tolerability, and Efficacy of MORAb-202 (Herein Referred to as Farletuzumab Ecteribulin), a Folate Receptor Alpha (FRα)-Targeting Antibody-drug Conjugate (ADC) in Participants With Selected Tumor Types

Is NCT04300556 recruiting? Yes, currently enrolling (May 2026). This Phase 1/2 trial studies multiple treatments for solid tumor.

Phase 1/2RecruitingEisai Inc.NCT04300556Data as of May 2026

Treatment: Farletuzumab ecteribulin · Prednisone · Prednisolone · Dexamethasone · LenvatinibThe primary objectives of the study are: (1) in the dose-escalation part: to evaluate safety and tolerability and to determine the recommended Phase 2 dose (RP2D) of farletuzumab ecteribulin (MORAb-202) in participants with selected tumor types (ovarian cancer \[OC\], endometrial cancer \[EC\], non-small cell lung carcinoma \[NSCLC\], triple-negative breast cancer \[TNBC\]), and (2) in dose-confirmation part: to evaluate preliminary efficacy measured by objective response rate (ORR) of farletuzumab ecteribulin (MORAb-202) in participants with OC and EC at selected doses and to further evaluate the safety and tolerability of farletuzumab ecteribulin (MORAb-202) and (3) dose-optimization part. (divided in two parts: Part A \[OC and EC participants\] and Part B \[OC only\]): Part A: to evaluate other farletuzumab ecteribulin (MORAb-202) treatment regimens for safety, tolerability and preliminary efficacy in participants with OC and EC; to evaluate the addition of short course of oral corticosteroids following every dose of farletuzumab ecteribulin (MORAb-202) administered every 21 days; and to select treatment regimens with farletuzumab ecteribulin (MORAb-202) for further evaluation in Part B. Part B: to evaluate the safety and tolerability of different doses of farletuzumab ecteribulin (MORAb-202) as monotherapy and in combination with lenvatinib and to determine the recommended dose (RD) of farletuzumab ecteribulin (MORAb-202) as monotherapy and in combination with lenvatinib.

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Extracted eligibility criteria

Cancer type

Tumor Agnostic

Biomarker criteria

Required: FOLR1 any tested (testing required; no minimum expression threshold)

Available tumor tissue for FRA expression percent (%) by IHC analysis as assessed at a central laboratory. There is no minimum requirement for FRA expression (%).

Disease stage

Required: Stage IV

advanced, recurrent or metastatic

Performance status

ECOG 0–1(Restricted strenuous activity)

Prior therapy

Must have received: systemic anticancer therapy — metastatic

Previously treated with at least one line of systemic anticancer therapy (cytotoxic or targeted anticancer agents) in the metastatic setting. [TNBC]

Must have received: systemic therapy — metastatic

participants who have failed previous treatment for metastatic disease [NSCLC adenocarcinoma]

Must have received: platinum-based regimen or immunotherapy-based regimen

Relapsed or failure of at least one platinum-based regimen or one immunotherapy-based regimen [EC]

Must have received: platinum-containing chemotherapy

platinum-resistant disease (defined as progression within 6 months after the last dose of at least 4 cycles of the last platinum containing chemotherapy regimen) [OC/primary peritoneal/fallopian tube cancer]

Cannot have received: folate receptor targeting agents

Exception: mirvetuximab soravtansine in the setting of FRA >=75%

Participants who received previous treatment with any folate receptor targeting agents, except for mirvetuximab soravtansine in the setting of FRA >=75%

Cannot have received: chest radiotherapy

Exception: chest wall radiation > 2 years before starting study treatment

History of chest radiotherapy. Participants with history of chest wall radiation (example, history of breast cancer) may be permitted if chest wall radiation is documented > 2 years before starting study treatment.

Cannot have received: pneumonectomy

Prior pneumonectomy

Lab requirements

Blood counts

ANC >=1.0*10^9/L (MORAb-202 monotherapy); ANC >=1.5*10^9/L (MORAb-202 plus lenvatinib); Hgb >=9.0 g/dL; Platelet count >=75*10^9/L

Kidney function

Serum creatinine <=1.5 mg/dL or calculated creatinine clearance >=50 mL/min (Cockcroft-Gault formula for Dose Optimization Part B)

Liver function

Total bilirubin <=1.5*ULN except for unconjugated hyperbilirubinemia (e.g., Gilbert's syndrome); ALT and AST <=3*ULN (<=5*ULN with liver metastases); ALP <=3*ULN unless known bone metastases; Albumin >3.0 g/dL

Adequate renal function as evidenced by serum creatinine <=1.5 mg/dL or calculated creatinine clearance >=50 mL/min... Adequate bone marrow function... Adequate liver function...

Structured fields extracted by AI. May contain errors — verify against the official protocol.

US trial sites

  • ACRC/Arizona Clinical Research Center, Inc · Tucson, Arizona
  • Universty of Arkansas for Medical Sciences · Little Rock, Arkansas
  • Stanford Women's Cancer Center · Palo Alto, California
  • University of Miami · Coral Gables, Florida
  • Moffitt Cancer Center and Research Institute · Tampa, Florida

Showing up to 5 US sites. See all sites on ClinicalTrials.gov →

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