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OncoMatch/Clinical Trials/NCT03816319

TAK-243 in Treating Patients With Relapsed or Refractory Acute Myeloid Leukemia or Myelodysplastic Syndromes With Increased Blasts

Is NCT03816319 recruiting? Yes, currently enrolling (Aug 2026). This Phase 1 trial studies UAE Inhibitor TAK-243 for myelodysplastic syndrome with excess blasts.

Phase 1RecruitingNational Cancer Institute (NCI)NCT03816319Data as of Aug 2026Location: United States · Canada

Treatment: UAE Inhibitor TAK-243This phase I trial studies the side effects and best dose of TAK-243 in treating patients with acute myeloid leukemia or myelodysplastic syndromes with increased blasts that has come back (relapsed) or that is not responding to treatment (refractory). TAK-243 may stop the growth of cancer cells by blocking some of the enzymes needed for cell growth.

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Extracted eligibility criteria

Treatments studied

Other

UAE Inhibitor TAK-243

Cancer type

Myelodysplastic Syndrome

Acute Myeloid Leukemia

Performance status

ECOG 0–2(Ambulatory, capable of self-care)

Prior therapy

Min 1 prior line

Must have received: systemic therapy — relapsed or refractory AML or MDS-IB

Patients must have relapsed or refractory disease after receiving at least one prior line of therapy

Lab requirements

Kidney function

Serum creatinine < 176 mcmol/L (2 mg/dL) OR creatinine clearance ≥ 60 mL/min (Cockcroft-Gault)

Liver function

Serum bilirubin <= 1.5 × institutional ULN (Gilbert's syndrome allowed); AST/ALT <= 3 × institutional ULN

Cardiac function

Documented normal cardiac function (>= 50%) by echocardiogram or MUGA scan

Serum bilirubin <= 1.5 × institutional ULN (Gilbert's syndrome allowed); AST/ALT <= 3 × institutional ULN; Serum creatinine < 176 mcmol/L (2 mg/dL) OR creatinine clearance ≥ 60 mL/min (Cockcroft-Gault); Documented normal cardiac function (>= 50%) by echocardiogram or MUGA scan

Structured fields extracted by AI. May contain errors — verify against the official protocol.

US trial sites

  • Moffitt Cancer Center · Tampa, Florida
  • Northwestern University · Chicago, Illinois
  • Ohio State University Comprehensive Cancer Center · Columbus, Ohio
  • VCU Massey Comprehensive Cancer Center · Richmond, Virginia

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See all sites on ClinicalTrials.gov →

Frequently asked questions

Is NCT03816319 currently recruiting?

Yes, this trial is currently recruiting patients.

Is prior treatment required for enrollment?

Yes. Patients must have previously received systemic therapy.

Could you qualify for this trial?

Enter your biomarker results to see how this trial's eligibility criteria match your specific cancer profile.

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